{"title":"Protein Kinases","description":"\u003ch3 class=\"highlited\"\u003e\u003cspan\u003eAbout Protein kinases:\u003c\/span\u003e\u003c\/h3\u003e\n\u003cp\u003eProtein kinases are a group of kinase enzymes found within the human body. The list of roughly 500 protein kinase genes make up about 2% of human genes. The enzymes alter other proteins through a process known as phosphorylation, which is where phosphate groups are added to them.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eProtein Kinase Structure\u003c\/strong\u003e\u003cbr\u003eProtein kinases are enzymes located in the cytoplasm that phosphorylates proteins. The chief enzymes consist of PKA, PKG, PKC, and tyrosyl protein kinases. The eukaryotic protein kinases belong to a wide and varied family of proteins that boast a shared conserved catalytic core. The N-terinal of the catalytic domain contains glycine residues close to the lysine amino aid, having an influence on ATP binding Meanwhile, the central region of the catalyic domain has a conserved aspartic acid.\u003cbr\u003ePhosphorylation of the proteins is very quick due to the rapid dephosphorylate of previously phosphorylated cells, resulting in the termination of the intracellular signal. By regulating the biological activity of proteins, the protein kinases induce a change from inactivity to activity within the target cells.\u003cbr\u003eExamples of human proteins including the protein kinase domain include but are not limited to; AAK1, AATK, ARAF, AURKA, AXL, BLK, BMPR1A, BMPR1B, BMX, CAMK4, CDK1, CDK10, CHUK, CIT, DYRK1A, DYRK1B, EGFR, FER, FES, GAK, HUNK, IT, KSR1, KSR2, LCK, LIMK1, LIMK2, MAP2K5, MYLK4, NRK, OXRS1, PLK1, PLK2, POMK, RET, ROCK1, ROCk2, SIK1, SIK2, LK, TEC, TEK, ULK1, ULK2, WEE1, and ZAP70.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eProtein Kinase Function and Mechanisms\u003c\/strong\u003e\u003cbr\u003eAs the largest enzyme superfamily related to cell signal transduction, protein kinases are therapeutic targets for various diseases. Protein kinases can, through phosphorylation, alter protein functions in several ways. It may increase or decrease the protein’s activity, stabilize it, or even lead to its destruction.\u003cbr\u003eThe enzymes can also localize the protein while regulating the enzyme too. Because it is a reversible covalent modifications, prosphorylation is seen to be regulatory. Allosteric control, for example, responds to signals outside of the cell. The phosphorylation is more frequent in eukaryotic cells than prokaryotic cells due to their wider response rate.\u003cbr\u003ePathways affected by protein kinases include metabolism, cell signalling, protein regulation, cellular transport, secretory processes. Protein kinases will influence both activity and reactivity, as well as binding mechanisms in relation to other molecules.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eProtein Kinase Interactions\u003c\/strong\u003e\u003cbr\u003eRoughly 30% of all human proteins can be changed by the protein kinase activities, affecting signal transduction and other cellular pathways. The majority act on both serine and theonine while others interact with tyrosine. Dual-specificity kinases act on all three.Kinases are turned on or off by phosphorylation, having huge impact on the target cell.\u003cbr\u003eThe serine and theonine protein kinases phosphorylate the OH group and may be regulated by various events such as DNA damage, as well as chemical signals such as cAMP\/cGMP, diacylglycerol, and Ca2+\/calmodulin.\u003cbr\u003eAnother significant group of protein kinases is the mitogen-activated protein (MAP) kinases. protein phosphatases can limit the activity on the MAP kinases while the activation of transmembrane receptors via natural ligands or crosslinking agents send signals that include oxidant stress.\u003c\/p\u003e","products":[{"product_id":"mertk-mouse","title":"MERTK Mouse","description":"\u003cp\u003eMER Proto-Oncogene Tyrosine Kinase Mouse Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eTyrosine-protein kinase Mer, Proto-oncogene c-Mer, Receptor tyrosine kinase MerTK, Mertk, 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Kinase.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"2µg","offer_id":43173938495572,"sku":"PKA-062","price":60.0,"currency_code":"USD","in_stock":true},{"title":"10µg","offer_id":43173938528340,"sku":"PKA-062","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43173938561108,"sku":"PKA-062","price":5200.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-csk-human-PKA-062.png?v=1776441085"},{"product_id":"acka-ecoli","title":"ACKA E.Coli","description":"\u003cp\u003eAcetate Kinase E.Coli Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eAcetate kinase, Acetokinase, ackA, ack, ACKA, Acetate kinase A and propionate kinase 2.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"5µg","offer_id":43173944590420,"sku":"PKA-063","price":60.0,"currency_code":"USD","in_stock":true},{"title":"20µg","offer_id":43173944623188,"sku":"PKA-063","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43173944655956,"sku":"PKA-063","price":2700.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-acka-ecoli-PKA-063.png?v=1776676369"},{"product_id":"mob1b-human","title":"MOB1B Human","description":"\u003cp\u003eMOB Kinase Activator 1B Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eMOB\nKinase Activator 1B, Mps One Binder Kinase Activator-Like 1A, Mob1 Homolog 1A, MOBKL1A,\nMob1A, MOB4A, MOB1, Mps One Binder Kinase Activator-Like 1A (Yeast), MOB1, Mps\nOne Binder Kinase Activator-Like 1A, MOB1 Mps One Binder Homolog B (Yeast), MOB1\nMps One Binder Homolog B, Mob4A Protein, MATS2, Mob1B, MOB kinase activator 1B.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"5µg","offer_id":43174031720532,"sku":"PKA-054","price":60.0,"currency_code":"USD","in_stock":true},{"title":"20µg","offer_id":43174031753300,"sku":"PKA-054","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174031786068,"sku":"PKA-054","price":2700.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-mob1b-human-PKA-054.png?v=1776444236"},{"product_id":"mob3b-human","title":"MOB3B Human","description":"\u003cp\u003eMOB Kinase Activator 3B Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eMOB Kinase Activator 3B, Chromosome 9 Open Reading Frame 35, Monopolar Spindle 1 Binding, MOB1, Domain Containing, MOB1 Mps One Binder Kinase Activator-Like 2B, Mps One Binder Kinase Activator-Like 2B, Monopolar Spindle 1 Binding, Mob1 Homolog 2b, MOBKL2B, Domain Containing, C9orf35, MOB1D, MOB1.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"2µg","offer_id":43174032670804,"sku":"PKA-319","price":60.0,"currency_code":"USD","in_stock":true},{"title":"10µg","offer_id":43174032703572,"sku":"PKA-319","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174032736340,"sku":"PKA-319","price":5200.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-mob3b-human-PKA-319.png?v=1776702706"},{"product_id":"akap7-human","title":"AKAP7 Human","description":"\u003cp\u003eA Kinase Anchor Protein 7 Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eA kinase (PRKA) anchor protein 7, A-kinase anchor protein 18 kDa, A-kinase anchor protein 9, kDa PRKA7 isoforms alpha\/beta, PRKA7 isoform gamma, AKAP15, AKAP18.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"2µg","offer_id":43174068355156,"sku":"PKA-030","price":60.0,"currency_code":"USD","in_stock":true},{"title":"10µg","offer_id":43174068387924,"sku":"PKA-030","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174068420692,"sku":"PKA-030","price":5200.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-akap7-human-PKA-030.png?v=1776440210"},{"product_id":"dck-human","title":"DCK Human","description":"\u003cp\u003eDeoxycytidine Kinase Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eDeoxycytidine kinase, DCK, MGC117410, MGC138632.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"5µg","offer_id":43174081134676,"sku":"PKA-313","price":60.0,"currency_code":"USD","in_stock":true},{"title":"20µg","offer_id":43174081167444,"sku":"PKA-313","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174081200212,"sku":"PKA-313","price":3600.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-dck-human-PKA-313.png?v=1776441655"},{"product_id":"akt3-human","title":"AKT3 Human","description":"\u003cp\u003eAKT Serine\/Threonine Kinase 3 Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eRAC-gamma serine\/threonine-protein kinase, Protein kinase Akt-3, Protein kinase B gamma, PKB gamma, RAC-PK-gamma, STK-2, AKT3, PKBG.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"5µg","offer_id":43174087032916,"sku":"PKA-130","price":60.0,"currency_code":"USD","in_stock":true},{"title":"20µg","offer_id":43174087065684,"sku":"PKA-130","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174087098452,"sku":"PKA-130","price":3600.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-akt3-human-PKA-130.png?v=1776440298"},{"product_id":"mvk-human","title":"MVK Human","description":"\u003cp\u003eMevalonate Kinase Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eMevalonate Kinase (Mevalonic Aciduria), LH Receptor MRNA-Binding Protein, LRBP, Mevalonate Kinase 1, MK, MVLK, EC 2.7.1.36.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"5µg","offer_id":43174104236116,"sku":"PKA-052","price":60.0,"currency_code":"USD","in_stock":true},{"title":"20µg","offer_id":43174104268884,"sku":"PKA-052","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174104301652,"sku":"PKA-052","price":2700.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-mvk-human-PKA-052.png?v=1776444479"},{"product_id":"nagk-human","title":"NAGK Human","description":"\u003cp\u003eN-Acetylglucosamine Kinase Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eN-acetylglucosamine kinase, GNK, GlcNAc kinase, N-acetyl-D-glucosamine kinase, HSA242910, EC 2.7.1.59.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"5µg","offer_id":43174154207316,"sku":"PKA-027","price":60.0,"currency_code":"USD","in_stock":true},{"title":"20µg","offer_id":43174154240084,"sku":"PKA-027","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174154272852,"sku":"PKA-027","price":2700.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-nagk-human-PKA-027.png?v=1776444659"},{"product_id":"sgk1-human","title":"SGK1 Human","description":"\u003cp\u003eSerum\/Glucocorticoid Regulated Kinase 1 Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eSerine\/threonine-protein kinase Sgk1, Serum\/glucocorticoid-regulated kinase 1, SGK1, SGK.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"2µg","offer_id":43174181404756,"sku":"PKA-272","price":60.0,"currency_code":"USD","in_stock":true},{"title":"10µg","offer_id":43174181437524,"sku":"PKA-272","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174181470292,"sku":"PKA-272","price":5200.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-sgk1-human-PKA-272.png?v=1776445808"},{"product_id":"ndk-ecoli","title":"NDK E.Coli","description":"\u003cp\u003eNucleoside Diphosphate Kinase E.Coli Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eNucleoside diphosphate kinase, NDK, NDP kinase, Nucleoside-2-P kinase, b2518, JW2502.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"5µg","offer_id":43174202769492,"sku":"PKA-034","price":60.0,"currency_code":"USD","in_stock":true},{"title":"20µg","offer_id":43174202802260,"sku":"PKA-034","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174202835028,"sku":"PKA-034","price":2700.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-ndk-ecoli-PKA-034.png?v=1776703068"},{"product_id":"nek7-human","title":"NEK7 Human","description":"\u003cp\u003eNIMA-related kinase 7 Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eNIMA (never in mitosis gene a)-related kinase 7, Serine\/threonine-protein kinase 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kinase.\u003c\/p\u003e\n\u003c\/div\u003e","brand":"prospecbio","offers":[{"title":"5µg","offer_id":43174236684372,"sku":"PKA-005","price":60.0,"currency_code":"USD","in_stock":true},{"title":"20µg","offer_id":43174236717140,"sku":"PKA-005","price":145.0,"currency_code":"USD","in_stock":true},{"title":"1mg","offer_id":43174236749908,"sku":"PKA-005","price":2700.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0559\/3219\/0804\/files\/Prospecbio-dtymk-human-PKA-005.png?v=1776682918"},{"product_id":"skp1-human","title":"SKP1 Alpha Human","description":"\u003cp\u003eS-phase Kinase-Associated Protein 1 Isoform A Human Recombinant\u003c\/p\u003e\n\n\u003cdiv class=\"synonyms_hide\"\u003e\n  \u003cp\u003eSKP-1, EMC19, MGC34403, OCP-II, OCP2, p19A, SKP1A, TCEB1L, S-phase kinase-associated protein 1, Cyclin-A\/CDK2-associated protein p19, p19skp1, RNA polymerase II elongation factor-like protein, Organ of Corti protein 2, OCP-2, Organ of Corti 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